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Eliquis
Anticoagulant • Direct factor Xa inhibitor
PremiumHalf-life
12 h
Protein Binding
Metabolized By
CYP3A4, CYP1A2, CYP2A6, CYP2B6, CYP2C8, CYP2C9, CYP2D6, CYP2C19
External
Drugs.comDirectly inhibits factor Xa, reducing thrombin generation
Drug Class
Anticoagulant
Subclass
Direct factor Xa inhibitor
Half-life
12 h
Time for plasma concentration to decrease by 50%
Protein Binding
—
Fraction bound to plasma proteins
Therapeutic Index
Wide
Margin between therapeutic and toxic doses