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Topamax, Trokendi XR, Qudexy XR, Qsymia, Trokendi, Qudexy, Eprontia
Antiepileptic • Sulfamate-substituted monosaccharide
PremiumMultiple: blocks Na+ channels, enhances GABA, inhibits glutamate, weak carbonic anhydrase inhibitor
Drug Class
Antiepileptic
Subclass
Sulfamate-substituted monosaccharide
Half-life
21 hours
Time for plasma concentration to decrease by 50%
Protein Binding
—
Fraction bound to plasma proteins
Therapeutic Index
Wide
Margin between therapeutic and toxic doses