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Plaquenil
DMARD • Antimalarial / Immunomodulator
Accumulates in lysosomes, raising pH and inhibiting antigen presentation; reduces cytokine production
Drug Class
DMARD
Subclass
Antimalarial / Immunomodulator
Half-life
40-50 days
Time for plasma concentration to decrease by 50%
Protein Binding
45%
Fraction bound to plasma proteins
Therapeutic Index
Wide
Margin between therapeutic and toxic doses